What is the catalog number for Cobimetinib (GDC-0973)?

The catalog number for Cobimetinib (GDC-0973) is C13147-10mM/1mL.

What sizes are available for Cobimetinib (GDC-0973)?

Cobimetinib (GDC-0973) is available in the following size(s): 10 mM/1mL.

Is Cobimetinib (GDC-0973) in stock?

Cobimetinib (GDC-0973) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Cobimetinib (GDC-0973)?

Cobimetinib (GDC-0973) is requires dry ice shipping.

Cobimetinib (GDC-0973)

Product Specifications

CAS Number

934660-93-2

Synonyms

RG7420, XL518

Target

MEK

Applications

Protein Tyrosine Kinase

Smiles

C1CCNC (C1) C2 (CN (C2) C (=O) C3=C (C (=C (C=C3) F) F) NC4=C (C=C (C=C4) I) F) O

Molecular Formula

C21H21F3IN3O2

Additionnal Information

Cobimetinib (GDC-0973, RG7420) is a potent and highly selective MEK1 inhibitor with IC50 of 4.2 nM, and showing no significant inhibition when tested against a panel of more than 100 of serine-threonine and tyrosine kinases. Cobimetinib induces apoptosis. Phase 3.