UPF 1069
Product Specifications
CAS Number
1048371-03-4
Target
PARP
Applications
DNA Damage/DNA Repair
Smiles
C1=CC=C (C=C1) C (=O) COC2=CC=CC3=C2C=CNC3=O
Molecular Formula
C17H13NO3
Additionnal Information
UPF 1069 is a selective PARP2 inhibitor with IC50 of 0.3 μM. It is ~27-fold selective against PARP1.
Storage Conditions
2 years -80 in solvent
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