GSK864
Product Specifications
CAS Number
1816331-66-4
Target
Dehydrogenase
Applications
Metabolism
Molecular Formula
C30H31FN6O4
Additionnal Information
GSK864 is a cell-penetrant, potent, and selective inhibitor of isocitrate dehydrogenase 1 (IDH1) mutants, specifically targeting the R132C, R132H, and R132G variants with IC50 values of 8.8 nM, 15.2 nM, and 16.6 nM, respectively.
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