What is the catalog number for Pelabresib (CPI-0610)?

The catalog number for Pelabresib (CPI-0610) is C13001-100mg.

What sizes are available for Pelabresib (CPI-0610)?

Pelabresib (CPI-0610) is available in the following size(s): 100 mg.

Is Pelabresib (CPI-0610) in stock?

Pelabresib (CPI-0610) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Pelabresib (CPI-0610)?

Pelabresib (CPI-0610) is requires dry ice shipping.

Pelabresib (CPI-0610)

Product Specifications

CAS Number

1380087-89-7

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CC1=NOC2=C1C3=CC=CC=C3C (=NC2CC (=O) N) C4=CC=C (C=C4) Cl

Molecular Formula

C20H16ClN3O2

Additionnal Information

Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.