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Bufalin

Product Specifications

CAS Number

465-21-4

Synonyms

BF

Target

ATPase

Applications

Transmembrane Transporters

Molecular Formula

C24H34O4

Additionnal Information

Bufalin (BF) is a potent inhibitor of steroid receptor coactivator SRC-3, SRC-1 and Na+/K+-ATPase. Bufalin binds to the subunit α1, α2 and α3 of Na+/K+-ATPase with Kd of 42.5 nM, 45 nM and 40 nM, respectively. Bufalin is a major immunoreactive component isolated from the Chinese medicine Chan Su with anti-cancer activity.

Storage Conditions

3 years -20°C powder

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