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MI-136

Product Specifications

CAS Number

1628316-74-4

Target

Histone Methyltransferase

Applications

Epigenetics

Smiles

C1CN (CCC1NC2=C3C=C (SC3=NC=N2) CC (F) (F) F) CC4=CC5=C (C=C4) NC (=C5) C#N

Molecular Formula

C23H21F3N6S

Additionnal Information

MI-136 can specifically inhibit the menin-MLL interaction. It inhibits DHT-induced expression of androgen receptor (AR) target genes.

Storage Conditions

2 years -80 in solvent

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