What is the catalog number for Gilteritinib (ASP2215)?

The catalog number for Gilteritinib (ASP2215) is C12921-5mg.

What sizes are available for Gilteritinib (ASP2215)?

Gilteritinib (ASP2215) is available in the following size(s): 5 mg.

Is Gilteritinib (ASP2215) in stock?

Gilteritinib (ASP2215) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Gilteritinib (ASP2215)?

Gilteritinib (ASP2215) is requires dry ice shipping.

Gilteritinib (ASP2215)

Product Specifications

CAS Number

1254053-43-4

Target

FLT3

Applications

Protein Tyrosine Kinase

Smiles

CCC1=C (N=C (C (=N1) C (=O) N) NC2=CC (=C (C=C2) N3CCC (CC3) N4CCN (CC4) C) OC) NC5CCOCC5

Molecular Formula

C29H44N8O3

Additionnal Information

Gilteritinib (ASP2215) is a small-molecule FLT3/AXL inhibitor with IC50 values of 0.29 nM and 0.73 nM for FLT3 and AXL, respectively. It inhibits FLT3 at an IC50 value that was approximately 800-fold more potent than the concentration required to inhibit c-KIT (230 nM) .