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LFM-A13

Product Specifications

CAS Number

244240-24-2

Target

BTK

Applications

Protein Tyrosine Kinase

Smiles

CC (=C (C#N) C (=O) NC1=C (C=CC (=C1) Br) Br) O

Molecular Formula

C11H8Br2N2O2

Additionnal Information

LFM-A13 is a specific Bruton's tyrosine kinase (BTK) inhibitor with IC50 of 2.5 μM, >100-fold selectivity over other protein kinases including JAK1, JAK2, HCK, EGFR, and IRK.

Storage Conditions

2 years -80 in solvent

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