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Sotuletinib (BLZ945)

Product Specifications

CAS Number

953769-46-5

Target

CSF-1R

Applications

Protein Tyrosine Kinase

Smiles

CNC (=O) C1=NC=CC (=C1) OC2=CC3=C (C=C2) N=C (S3) NC4CCCCC4O

Molecular Formula

C20H22N4O3S

Additionnal Information

Sotuletinib (BLZ945) is an orally active, potent and selective CSF-1R inhibitor with IC50 of 1 nM, >1000-fold selective against its closest receptor tyrosine kinase homologs.

Storage Conditions

2 years -80 in solvent

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