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GDC-0623

Product Specifications

CAS Number

1168091-68-6

Synonyms

G-868

Target

MEK

Applications

Protein Tyrosine Kinase

Smiles

C1=CC (=C (C=C1I) F) NC2=C (C=CC3=CN=CN32) C (=O) NOCCO

Molecular Formula

C16H14FIN4O3

Additionnal Information

GDC-0623 (G-868) is a potent and ATP-uncompetitive MEK1 inhibitor with Ki of 0.13 nM. Phase 1.

Storage Conditions

2 years -80 in solvent

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