RS-102895 Hydrochloride
Product Specifications
CAS Number
1173022-16-6
Synonyms
RS-102895 HCl
Target
CCR
Applications
GPCR & G Protein
Smiles
Cl.FC (F) (F) C1=CC=C (CCN2CCC3 (CC2) OC (=O) NC4=CC=CC=C34) C=C1
Molecular Formula
C21H22ClF3N2O2
Additionnal Information
RS-102895 hydrochloride (HCl) is a potent antagonist of Chemokine (C-C motif) receptor 2 (CCR2) with IC50 of 360 nM, and shows no effect on CCR1. RS-102895 hydrochloride also inhibits human α1a and α1d receptors, rat brain cortex 5-HT1a receptor in cells with IC50s of 130 nM, 320 nM, 470 nM, respectively.
Storage Conditions
3 years -20°C powder
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