Apabetalone (RVX-208)
Product Specifications
CAS Number
1044870-39-4
Synonyms
RVX-000222
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1=CC (=CC (=C1OCCO) C) C2=NC3=C (C (=CC (=C3) OC) OC) C (=O) N2
Molecular Formula
C20H22N2O5
Additionnal Information
Apabetalone (RVX-208, RVX-000222) is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2 in a cell-free assay, about 170-fold selectivity over BD1. Phase 2.
Storage Conditions
2 years -80 in solvent
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