What is the catalog number for Molibresib (I-BET-762)?

The catalog number for Molibresib (I-BET-762) is C12512-50mg.

What sizes are available for Molibresib (I-BET-762)?

Molibresib (I-BET-762) is available in the following size(s): 50 mg.

Is Molibresib (I-BET-762) in stock?

Molibresib (I-BET-762) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Molibresib (I-BET-762)?

Molibresib (I-BET-762) is requires dry ice shipping.

Molibresib (I-BET-762)

Product Specifications

CAS Number

1260907-17-2

Synonyms

GSK525762, GSK525762A

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CCNC (=O) CC1C2=NN=C (N2C3=C (C=C (C=C3) OC) C (=N1) C4=CC=C (C=C4) Cl) C

Molecular Formula

C22H22ClN5O2

Additionnal Information

Molibresib (I-BET-762, GSK525762, GSK525762A) is an inhibitor for BET proteins with IC50 of ~35 nM in a cell-free assay, suppresses the production of proinflammatory proteins by macrophages and blocks acute inflammation, highly selective over other bromodomain-containing proteins.