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KPT-185

Product Specifications

CAS Number

1333151-73-7

Target

CRM1

Applications

Transmembrane Transporters

Smiles

CC (C) OC (=O) C=CN1C=NC (=N1) C2=CC (=CC (=C2) OC) C (F) (F) F

Molecular Formula

C16H16F3N3O3

Additionnal Information

KPT-185 is a selective CRM1 inhibitor that induces growth inhibition and apoptosis in a panel of NHL cell lines with a median IC50 ~25 nM.

Storage Conditions

2 years -80 in solvent

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