What is the catalog number for Pinometostat (EPZ5676)?

The catalog number for Pinometostat (EPZ5676) is C12414-1g.

What sizes are available for Pinometostat (EPZ5676)?

Pinometostat (EPZ5676) is available in the following size(s): 1 g.

Is Pinometostat (EPZ5676) in stock?

Pinometostat (EPZ5676) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Pinometostat (EPZ5676)?

Pinometostat (EPZ5676) is requires dry ice shipping.

Pinometostat (EPZ5676)

Product Specifications

CAS Number

1380288-87-8

Target

Histone Methyltransferase

Applications

Epigenetics

Smiles

CC (C) N (CC1C (C (C (O1) N2C=NC3=C (N=CN=C32) N) O) O) C4CC (C4) CCC5=NC6=C (N5) C=C (C=C6) C (C) (C) C

Molecular Formula

C30H42N8O3

Additionnal Information

Pinometostat (EPZ5676) is an S-adenosyl methionine (SAM) competitive inhibitor of protein methyltransferase DOT1L with Ki of 80 pM in a cell-free assay, demonstrating >37,000-fold selectivity against all other PMTs tested, inhibits H3K79 methylation in tumor. Phase 1.