GSK126
Product Specifications
CAS Number
1346574-57-9
Synonyms
GSK2816126A, GSK2816126
Target
Histone Methyltransferase
Applications
Epigenetics
Smiles
CCC (C) N1C=C (C2=C (C=C (C=C21) C3=CN=C (C=C3) N4CCNCC4) C (=O) NCC5=C (C=C (NC5=O) C) C) C
Molecular Formula
C31H38N6O2
Additionnal Information
GSK126 (GSK2816126A, GSK2816126) is a potent, highly selective EZH2 methyltransferase inhibitor with IC50 of 9.9 nM, >1000-fold selective for EZH2 over 20 other human methyltransferases.
Storage Conditions
2 years -80 in solvent
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