GK921
Product Specifications
CAS Number
1025015-40-0
Target
Glutaminase
Applications
Proteases
Smiles
C1CCN (C1) CCOC2=NC3=C (N=CC=C3) N=C2C#CC4=CC=CC=C4
Molecular Formula
C21H20N4O
Additionnal Information
GK921 is a transglutaminase 2 (TGase 2) inhibitor with an IC50 of 8.93 μM under a modified assay condition.
Storage Conditions
3 years -20°C powder
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