GSK 5959
Product Specifications
CAS Number
901245-65-6
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CN1C2=C (C=C (C (=C2) NC (=O) C3=CC=CC=C3OC) N4CCCCC4) N (C1=O) C
Molecular Formula
C22H26N4O3
Additionnal Information
GSK5959 is a potent and selective BRPF1 bromodomain inhibitor with an IC50 of 80 nM and exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains.
Storage Conditions
3 years -20°C powder
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