GSK0660
Product Specifications
CAS Number
1014691-61-2
Target
PPAR
Applications
DNA Damage/DNA Repair
Smiles
COC1=C (C=CC (=C1) NC2=CC=CC=C2) NS (=O) (=O) C3=C (SC=C3) C (=O) OC
Molecular Formula
C19H18N2O5S2
Additionnal Information
GSK0660 is a potent PPARβ/δ antagonist with a pIC50 of 6.8 (binding assay IC50 = 155 nM; antagonist assay IC50 = 300 nM) and is nearly inactive on PPARα and PPARγ with IC50s above approximately 10 μM.
Storage Conditions
3 years -20°C powder
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