Imidafenacin
Product Specifications
CAS Number
170105-16-5
Synonyms
KRP-197, ONO-8025
Target
AChR
Applications
Neuronal Signaling
Smiles
CC1=NC=CN1CCC (C2=CC=CC=C2) (C3=CC=CC=C3) C (=O) N
Molecular Formula
C20H21N3O
Additionnal Information
Imidafenacin (KRP-197, ONO-8025) is a urinary antispasmodic of the anticholinergic class. It is a novel antimuscarinic agent with safety and efficacy, has been clinically used for the treatment of overactive bladder. Imidafenacin (KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors (IC50=4.13 nM) . IC50 value: 0.3 nM (M3) .
Storage Conditions
3 years -20°C powder
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