Tasimelteon
Product Specifications
CAS Number
609799-22-6
Synonyms
BMS 214778, VEC 162
Target
MT Receptor
Applications
Neuronal Signaling
Smiles
CCC (=O) NCC1CC1C2=C3CCOC3=CC=C2
Molecular Formula
C15H19NO2
Additionnal Information
Tasimelteon (BMS 214778, VEC 162) is a selective dual melatonin receptor (MT1/MT2) agonist with 2.1-4.4 times greater affinity for the MT2 receptor believed to mediate circadian rhythm phase-shifting (Ki = 0.0692 nM and Ki = 0.17 nM in NIH-3T3 and CHOeK1 cells, respectively), than for the MT1 receptor (Ki = 0.304 nM and Ki = 0.35 nM, respectively) .
Storage Conditions
3 years -20°C powder
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