TAK-285
Product Specifications
CAS Number
871026-44-7
Target
EGFR
Applications
Protein Tyrosine Kinase
Smiles
CC (C) (CC (=O) NCCN1C=CC2=C1C (=NC=N2) NC3=CC (=C (C=C3) OC4=CC=CC (=C4) C (F) (F) F) Cl) O
Molecular Formula
C26H25ClF3N5O3
Additionnal Information
TAK-285 is a novel dual HER2 and EGFR (HER1) inhibitor with IC50 of 17 nM and 23 nM, >10-fold selectivity for HER1/2 than HER4, less potent to MEK1/5, c-Met, Aurora B, Lck, CSK etc. Phase 1.
Storage Conditions
2 years -80 in solvent
More Discoveries
Explore Other Products
Browse additional items from our catalog
109A 11-80081 1 Each
Zipvap 8, 8 position evaporator for 28mm vials, insert heated only. Gas inlet not heated, with flowmeter. 115V
Sign In for Pricing
View Details 
MBS1402032-01 0.02 mg (E-Coli)
Recombinant Staphylococcus epidermidis 3-isopropylmalate dehydratase large subunit (leuC)
Sign In for Pricing
View Details 
MBS1402032-02 0.02 mg (Yeast)
Recombinant Staphylococcus epidermidis 3-isopropylmalate dehydratase large subunit (leuC)
Sign In for Pricing
View Details 
MBS1402032-03 0.1 mg (E-Coli)
Recombinant Staphylococcus epidermidis 3-isopropylmalate dehydratase large subunit (leuC)
Sign In for Pricing
View Details MBS1402032-04 0.1 mg (Yeast)
Recombinant Staphylococcus epidermidis 3-isopropylmalate dehydratase large subunit (leuC)
Sign In for Pricing
View Details MBS1402032-05 0.02 mg (Baculovirus)
Recombinant Staphylococcus epidermidis 3-isopropylmalate dehydratase large subunit (leuC)
Sign In for Pricing
View Details