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Mardepodect (PF-2545920)

Product Specifications

CAS Number

1292799-56-4

Target

PDE

Applications

Metabolism

Smiles

CN1C=C (C (=N1) C2=CC=C (C=C2) OCC3=NC4=CC=CC=C4C=C3) C5=CC=NC=C5

Molecular Formula

C25H20N4O

Additionnal Information

Mardepodect (PF-2545920) is a potent and selective PDE10A inhibitor with IC50 of 0.37 nM, with >1000-fold selectivity over the PDE.

Storage Conditions

2 years -80 in solvent

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