What is the catalog number for Buparlisib (BKM120)?

The catalog number for Buparlisib (BKM120) is C08388-5mg.

What sizes are available for Buparlisib (BKM120)?

Buparlisib (BKM120) is available in the following size(s): 5 mg.

Is Buparlisib (BKM120) in stock?

Buparlisib (BKM120) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Buparlisib (BKM120)?

Buparlisib (BKM120) is requires dry ice shipping.

Buparlisib (BKM120)

Product Specifications

CAS Number

944396-07-0

Synonyms

NVP-BKM120

Target

PI3K

Applications

PI3K/Akt/mTOR

Smiles

C1COCCN1C2=NC (=NC (=C2) C3=CN=C (C=C3C (F) (F) F) N) N4CCOCC4

Molecular Formula

C18H21F3N6O2

Additionnal Information

Buparlisib (BKM120, NVP-BKM120) is a selective PI3K inhibitor of p110α/β/δ/γ with IC50 of 52 nM/166 nM/116 nM/262 nM in cell-free assays, respectively. Reduced potency against VPS34, mTOR, DNAPK, with little activity to PI4Kβ. Buparlisib induces apoptosis. Phase 2.