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BIBF-0775

Product Specifications

CAS Number

334951-90-5

Target

TGF-beta/Smad

Applications

TGF-beta/Smad

Smiles

CCN (C) C (=O) C1=CC2=C (C=C1) C (=C (N2) O) C (=NC3=CC=C (C=C3) CN4CCCCC4) C5=CC=CC=C5

Molecular Formula

C31H34N4O2

Additionnal Information

BIBF-0775 is a selective inhibitor of transforming growth factor β Receptor I (TGFβRI, Alk5) with an IC50 of 34nM.

Storage Conditions

3 years -20°C powder

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