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Galunisertib (LY2157299)

Product Specifications

CAS Number

700874-72-2

Target

TGF-beta/Smad

Applications

TGF-beta/Smad

Smiles

CC1=NC (=CC=C1) C2=NN3CCCC3=C2C4=C5C=C (C=CC5=NC=C4) C (=O) N

Molecular Formula

C22H19N5O

Additionnal Information

Galunisertib (LY2157299) is a potent TGFβ receptor I (TβRI) inhibitor with IC50 of 56 nM in a cell-free assay. Phase 2/3.

Storage Conditions

2 years -80 in solvent

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