Idelalisib (CAL-101)
Product Specifications
CAS Number
870281-82-6
Synonyms
GS-1101
Target
PI3K
Applications
PI3K/Akt/mTOR
Smiles
CCC (C1=NC2=C (C (=CC=C2) F) C (=O) N1C3=CC=CC=C3) NC4=NC=NC5=C4NC=N5
Molecular Formula
C22H18FN7O
Additionnal Information
Idelalisib (CAL-101) is a selective p110δ inhibitor with IC50 of 2.5 nM in cell-free assays; shown to have 40- to 300-fold greater selectivity for p110δ than p110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR. Idelalisib also stimulates autophagy.
Storage Conditions
2 years -80 in solvent
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
![HACE1 Mouse Monoclonal Antibody [Clone ID: OTI2C7]](https://cdn.genprice.uk/products/937/68dd18bb061270361e908ab2/imageurl/cf810064.webp)
BNC882877-100 1x 100 µL
CD45RB (B-Cell Marker) (PTPRC/2877R), CF488A conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
LY420698 100 µg
LRRC14B (NM_001080478) Human Over-expression Lysate
Sign In for Pricing
View Details