Pelitinib (EKB-569)
Product Specifications
CAS Number
257933-82-7
Target
EGFR
Applications
Protein Tyrosine Kinase
Smiles
CCOC1=C (C=C2C (=C1) N=CC (=C2NC3=CC (=C (C=C3) F) Cl) C#N) NC (=O) C=CCN (C) C
Molecular Formula
C24H23ClFN5O2
Additionnal Information
Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM. Pelitinib (EKB-569) also slightly inhibits Src, MEK/ERK and ErbB2 with IC50s of 282 nM, 800 nM and 1255 nM, respectively. Phase2.
Storage Conditions
2 years -80 in solvent
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