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TG100-115

Product Specifications

CAS Number

677297-51-7

Target

PI3K

Applications

PI3K/Akt/mTOR

Smiles

C1=CC (=CC (=C1) O) C2=NC3=C (N=C (N=C3N=C2C4=CC (=CC=C4) O) N) N

Molecular Formula

C18H14N6O2

Additionnal Information

TG100-115 is a PI3Kγ/δ inhibitor with IC50 of 83 nM/235 nM, with little effect on PI3Kα/β. Phase 1/2.

Storage Conditions

2 years -80 in solvent

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