GSK1904529A
Product Specifications
CAS Number
1089283-49-7
Synonyms
GSK 4529
Target
IGF-1R
Applications
Protein Tyrosine Kinase
Smiles
CCC1=CC (=C (C=C1N2CCC (CC2) N3CCN (CC3) S (=O) (=O) C) OC) NC4=NC=CC (=N4) C5=C (N=C6N5C=CC=C6) C7=CC (=C (C=C7) OC) C (=O) NC8=C (C=CC=C8F) F
Molecular Formula
C44H47F2N9O5S
Additionnal Information
GSK1904529A (GSK 4529) is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM in cell-free assays, >100-fold more selective for IGF-1R/InsR than Akt1/2, Aurora A/B, B-Raf, CDK2, EGFR etc.
Storage Conditions
2 years -80 in solvent
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC042430-500 1x 500 µL
YBX1 / Y-box Binding Protein 1 / YB-1 (Tumor Biomarker) (YBX1/2430), CF405S conjugate, 0.1mg/mL
Sign In for Pricing
View Details