BMS-536924
Product Specifications
CAS Number
468740-43-4
Synonyms
CS-0117
Target
IGF-1R
Applications
Protein Tyrosine Kinase
Smiles
CC1=CC (=CC2=C1N=C (N2) C3=C (C=CNC3=O) NCC (C4=CC (=CC=C4) Cl) O) N5CCOCC5
Molecular Formula
C25H26ClN5O3
Additionnal Information
BMS-536924 (CS-0117) is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.
Storage Conditions
2 years -80 in solvent
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