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MELK-8a Dihydrochloride

Product Specifications

CAS Number

1922153-17-0 (free base)

Target

MELK

Applications

PI3K/Akt/mTOR

Smiles

CN1CCN (CC1) C2=CC=C (C=C2) N3C=C (C=N3) C4=C (C=NC=C4) OCC5CCNCC5

Molecular Formula

C25H34Cl2N6O

Additionnal Information

MELK-8a Dihydrochloride is a novel inhibitor of maternal embryonic leucine zipper kinase (MELK) with an IC50 of 2 nM.

Storage Conditions

3 years -20°C powder

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