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LOC14

Product Specifications

CAS Number

877963-94-5

Target

PDI

Applications

ER stress & UPR

Smiles

C1CC1C (=O) N2CCN (CC2) CN3C (=O) C4=CC=CC=C4S3

Molecular Formula

C16H19N3O2S

Additionnal Information

LOC14 is a potent inhibitor of protein disulfide isomerase (PDI) with EC50 of 500 nM and Kd of 62 nM, respectively.

Storage Conditions

3 years -20°C powder

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