Amezalpat
Product Specifications
CAS Number
1616372-41-8
Synonyms
TPST-1120
Additionnal Information
Amezalpat is a first-in-class, oral, competitive antagonist of peroxisome proliferator-activated receptor α (PPARα), with IC50 of 0.04 μM. It inhibits fatty acid oxidation (FAO), disrupting cancer cell metabolism and restoring immune responses, and shows antitumor activity in research on advanced solid tumors.
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