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PIM447

Product Specifications

CAS Number

1210608-43-7

Synonyms

LGH447

Additionnal Information

PIM447 (LGH447) is a potent, orally available, and selective pan-PIM kinase inhibitor, with Ki values of 6, 18, and 9 pM for PIM1, PIM2, and PIM3, respectively. PIM447 displays dual antimyeloma and bone-protective effects. PIM447 induces apoptosis.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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