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UNC0321

Product Specifications

CAS Number

1238673-32-9

Target

G9a/GLP

Applications

Epigenetics

Molecular Formula

C27H45N7O3

Additionnal Information

UNC0321 is a potent and selective inhibitor of G9a histone methyltransferase. It displays high potency at the picomolar level, with a Ki of 63 pM and assay-dependent IC50 values between 6-9 nM. UNC0321 also acts as an inhibitor of GLP. It demonstrates anti-apoptotic effects and holds potential for therapeutic use in diabetic vascular complications.

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