Darifenacin
Product Specifications
CAS Number
133099-04-4
Synonyms
UK-88525
Target
AChR
Applications
Neuronal Signaling
Molecular Formula
C28H30N2O2
Additionnal Information
Darifenacin (UK-88525) is a selective and orally active antagonist of M3 muscarinic receptor (M3R) with a pKi of 8.86. It exhibits efficacy in overactive bladder, partly due to bladder afferent desensitization. It also shows potential in preventing liver injury and inhibiting colorectal cancer growth in both in vitro and in vivo models.
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