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Talmapimod

Product Specifications

CAS Number

309913-83-5

Synonyms

SCIO-469

Additionnal Information

Talmapimod (SCIO-469) is an orally active, selective, and ATP-competitive p38α inhibitor with an IC50 of 9 nM. Talmapimod shows about 10-fold selectivity over p38β, and at least 2000-fold selectivity over a panel of 20 other kinases, including other MAPKs.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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