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SSTC3

Product Specifications

CAS Number

1242422-09-8

Target

Casein Kinase

Applications

Cell Cycle

Molecular Formula

C23H17F3N4O3S2

Additionnal Information

SSTC3 is a potent activator of casein kinase 1α (CK1α) with a Kd of 32 nM that inhibits WNTsignaling with an EC50 of 30 nM. It attenuates CRC cell growth through CK1α-dependent WNT pathway inhibition, offering an improved therapeutic index for targeting WNT-driven tumors.

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