What is the catalog number for Phentolamine hydrochloride?

The catalog number for Phentolamine hydrochloride is C03693-5mg.

What sizes are available for Phentolamine hydrochloride?

Phentolamine hydrochloride is available in the following size(s): 5 mg.

Is Phentolamine hydrochloride in stock?

Phentolamine hydrochloride is currently made to order / not held in immediate stock. Contact us for lead time.

Phentolamine hydrochloride

Product Specifications

CAS Number

73-05-2

Target

Adrenergic Receptor

Applications

Neuronal Signaling

Molecular Formula

C17H19N3O.ClH

Additionnal Information

Phentolamine hydrochloride is a potent, selective, and orally active antagonist of α1 and α2 adrenergic receptors , with pKi values of 8.8, 8.0, and 8.3 for the human α2A, α2B, and α2C adrenergic receptors, respectively. It also shows binding affinities for the α1-adrenoceptor subtypes, exhibiting Ki values of 6.1 nM for cloned α1A/D, 39.8 nM for α1B, and 2.8 nM for α1C.