What is the catalog number for CP-100356 hydrochloride?

The catalog number for CP-100356 hydrochloride is C03651-100mg.

What sizes are available for CP-100356 hydrochloride?

CP-100356 hydrochloride is available in the following size(s): 100 mg.

Is CP-100356 hydrochloride in stock?

CP-100356 hydrochloride is currently made to order / not held in immediate stock. Contact us for lead time.

CP-100356 hydrochloride

Product Specifications

CAS Number

142715-48-8

Target

BCRP

Applications

Transmembrane Transporters

Molecular Formula

C31H36N4O6.ClH

Additionnal Information

CP-100356 hydrochloride is an orally active dual inhibitor of MDR1 (P-gp) and BCRP, with IC50 of ∼0.5 μM for MDR1-mediated calcein-AM transport inhibition and ∼1.5 μM for BCRP-mediated prazosin transport inhibition. It is also a weak inhibitor of OATP1B1 (IC50 ∼ 66 μM) .