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Ebio1

Product Specifications

CAS Number

339287-36-4

Target

Potassium Channel

Applications

Transmembrane Transporters

Molecular Formula

C19H14FNO

Additionnal Information

Ebio1 is a subtype-selective activator of the voltage-gated potassium channel KCNQ2 that enhances conductance through a unique twist-to-open mechanism. It induces conformational changes in the S6 helix, increasing channel activity at a saturating voltage (+50 mV) .

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