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DDD85646

Product Specifications

CAS Number

1215010-55-1

Synonyms

IMP-366

Molecular Formula

C21H24Cl2N6O2S

Additionnal Information

DDD85646 (IMP-366) is an orally active inhibitor of N-myristoyltransferase (NMT), with an IC50 of 2 nM for Trypanosoma brucei NMT (TbNMT) and 4 nM for human NMT (hNMT) . It exhibits a potential for treating human African trypanosomiasis.

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