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AZ3246

Product Specifications

CAS Number

2893978-54-4

Target

MAP4K

Applications

MAPK

Molecular Formula

C21H20F3N9O

Additionnal Information

AZ3246 is a selective inhibitor of HPK1 with an IC50 value of <3 nM. AZ3246 induces IL-2 secretion in T cells with an EC50 of 90 nM and demonstrates antitumor activity in in vivo models.

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