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Wu-5

Product Specifications

CAS Number

2630378-05-9

Target

DUB

Applications

Ubiquitin

Molecular Formula

C15H13NO7S

Additionnal Information

Wu-5 is an inhibitor of USP10 that blocks its activity in vitro with an IC50 of 8.3 μM. It also promotes FLT3-ITD degradation and synergistically enhances crenolanib-induced apoptosis.

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