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PDK4-IN-1 hydrochloride

Product Specifications

CAS Number

2310262-11-2

Target

Dehydrogenase

Applications

Metabolism

Molecular Formula

C22H19N3O2.ClH

Additionnal Information

PDK4-IN-1 hydrochloride is an anthraquinone-derived, orally active allosteric inhibitor of PDK4 with an IC50 of 84 nM, exhibiting anticancer activity by regulating cell proliferation, transformation, and apoptosis. It also exhibit antidiabeti and anti-allergic activity.

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