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Lenumlostat

Product Specifications

CAS Number

2007885-39-2

Synonyms

PAT-1251; GB2064

Molecular Formula

C18H17F4N3O3

Additionnal Information

Lenumlostat (PAT-1251, GB2064) is a potent, selective, and orally available inhibitor of lysyl oxidase-like 2 (LOXL2) . It exhibits greater selectivity for LOXL2 over other family members, with IC50 of 0.71 μM for hLOXL2 and 1.17 μM for hLOXL3. It also possesses anti-fibrotic properties.

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