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Sevasemten

Product Specifications

CAS Number

2417395-15-2

Synonyms

EDG-5506

Target

MLCK

Applications

Cytoskeletal Signaling

Molecular Formula

C16H11F4N5O2

Additionnal Information

Sevasemten is a selective, orally active allosteric inhibitor of skeletal muscle myosin that protects skeletal muscle from contraction-induced injury. Sevasemten reduces biomarkers of muscle damage and fibrosis, while enhancing muscle strength and functional activity in models of Duchenne muscular dystrophy.

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