Tegaserod

Product Specifications

CAS Number

145158-71-0

Target

5-HT Receptor

Applications

Neuronal Signaling

Molecular Formula

C16H23N5O

Additionnal Information

Tegaserod is an orally active agonist of serotonin receptor 4 (5-HT4R) and also acts as an antagonist of 5-HT2B receptor with pKi values of 7.5, 8.4, and 7.0 for human recombinant 5-HT2A, 5-HT2B, and 5-HT2C receptors, respectively. Tegaserod has anti-tumor activity and is used in the research of irritable bowel syndrome (IBS) .