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Oclacitinib

Product Specifications

CAS Number

1208319-26-9

Synonyms

PF-03394197

Target

JAK

Applications

Angiogenesis

Molecular Formula

C15H23N5O2S

Additionnal Information

Oclacitinib (PF-03394197), an inhibitor of JAK is highly potent at inhibiting JAK1 with an IC50 value of 10 nM, respectively. Oclacitinib is highly potent against the JAK1 enzyme, displaying a 1.8-fold selectivity for JAK1 vs. JAK2 and a 9.9-fold selectivity toward JAK1 vs. JAK3.
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